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Molecular basis of antibacterial activity of thiosemicarbazide-based compounds

2012/05/D/NZ7/02278

Keywords

Descriptors

  • NZ7_14: Farmacja, farmakoterapia, farmakologia

Panel

NZ7 – Diagnostic tools, therapies and public health: public health, epidemiology, environmental health risks and occupational medicine, medical ethics, drug discovery and therapies, pharmacology

Host institution

Uniwersytet Medyczny w Lublinie, Wydział Farmaceutyczny z Oddziałem Analityki Medycznej

Voivodeship: lubelskie

Other projects carried out by the institution »

Principal investigator (from the host institution)

dr hab. Agata Paneth

Number of co-investigators in the project: 2

Call

SONATA 3 – announced on 2012-03-15

Amount awarded
283 750 PLN
Project start date
2013-02-04
Project end date
2017-08-03
Project duration
54 months (the same as in the proposal)
Project status
Project settled

Information in the final report

Publication in academic press/journals (10)

  1. Molecular Properties Prediction, Docking Studies, and Antimicrobial Screening of 1,3,4-Thiadiazole and S-Triazole Derivatives

    Authors:
    Agata Siwek, Tomasz Plech, Joanna Stefańska, Paweł Stączek and Aleksandra Strzelczyk
    Academic press:
    Current Computer-Aided Drug Design (year: 2014, volume: 10, pages: 46095), Publisher: Bentham Science
    Status:
    Published
    DOI:
    10.2174/15734099113096660033 – link to the publication

  2. Conformational Preference of Potassium Salts of N-Acylhydrazinecarbodithioates with Antifungal Activity. Combined Experimental and Theoretical Approach ;

    Authors:
    Agata Siwek, Tomasz Plech, Nazar Trotsko, Urszula Kosikowska, Anna Malm, Katarzyna Dzitko, Piotr Paneth
    Academic press:
    Current Computer-Aided Drug Design (year: 2014, volume: 10, pages: 205-216), Publisher: Bentham Science
    Status:
    Published
    DOI:
    10.2174/1573409910666140521152701 – link to the publication

  3. Synthesis and antibacterial activity of 1,4-dibenzoylthiosemicarbazide derivatives

    Authors:
    Agata Paneth, Paweł Stączek, Tomasz Plech, Aleksandra Strzelczyk, Dominika Janowska, Joanna Stefańska, Katarzyna Dzitko, Monika Wujec, Szymon Kosiek, Piotr Paneth
    Academic press:
    Biomedicine & Pharmacotherapy (year: 2017, volume: 88, pages: 1235-1242), Publisher: Elsevier
    Status:
    Published
    DOI:
    10.1016/j.biopha.2017.02.001 – link to the publication

  4. Design, synthesis and biological evaluation of 4- benzoyl-1-dichlorobenzoylthiosemicarbazides as potent Gram-positive antibacterial agents

    Authors:
    Agata Paneth, Tomasz Plech, Barbara Kaproń, Dominika Hagel, Urszula Kosikowska, Edyta Kuśmierz, Katarzyna Dzitko, Piotr Paneth
    Academic press:
    Journal of Enzyme Inhibition & Medicinal Chemistry (year: 2016, volume: 31, pages: 434–440), Publisher: Taylor & Francis
    Status:
    Published
    DOI:
    10.3109/14756366.2015.1036050 – link to the publication

  5. Structure-activity relationship studies of microbiologically active thiosemicarbazides derived from hydroxybenzoic acid hydrazides

    Authors:
    Tomasz Plech, Agata Paneth, Barbara Kaproń, Urszula Kosikowska, Anna Malm, Aleksandra Strzelczyk, Paweł Stączek
    Academic press:
    Chemical Biology & Drug Design (year: 2014, volume: 85, pages: 315-325), Publisher: Wiley
    Status:
    Published
    DOI:
    10.1111/cbdd.12392 – link to the publication

  6. Synthesis, Characterization and Antimicrobial Activity of 4-benzoyl-1-(pyrazin-2-ylcarbonyl)-thiosemicarbazide

    Authors:
    Dominika Hagel, Agata Siwek, Tomasz Plech
    Academic press:
    Journal of Single Molecule Research (year: 2014, volume: 2, pages: 46186), Publisher: Sciknow
    Status:
    Published
    DOI:
    10.12966/jsmr.03.02.2014 – link to the publication

  7. 1,4-Disubstituted Thiosemicarbazide Derivatives are Potent Inhibitors of Toxoplasma gondii Proliferation

    Authors:
    Katarzyna Dzitko, Agata Paneth, Tomasz Plech, Jakub Pawełczyk, Paweł Stączek, Joanna Stefańska, Piotr Paneth
    Academic press:
    Molecules (year: 2014, volume: 19, pages: 9926-9943), Publisher: MDPI
    Status:
    Published
    DOI:
    10.3390/molecules19079926 – link to the publication

  8. Lipophilicity Studies on Thiosemicarbazide Derivatives

    Authors:
    Agata Paneth, Anna Hawrył, Tomasz Plech, Mirosław Hawrył, Ryszard Świeboda, Dominika Janowska, Monika Wujec, Piotr Paneth
    Academic press:
    Molecules (year: 2017, volume: 22, pages: 952), Publisher: MDPI
    Status:
    Published
    DOI:
    10.3390/molecules22060952 – link to the publication

  9. Biological evaluation and molecular modelling study of thiosemicarbazide derivatives as bacterial type IIA topoisomerases inhibitors

    Authors:
    Agata Paneth, Paweł Stączek, Tomasz Plech, Aleksandra Strzelczyk, Katarzyna Dzitko, Monika Wujec, Edyta Kuśmierz, Urszula Kosikowska, Agnieszka Grzegorczyk, Piotr Paneth
    Academic press:
    Journal of Enzyme Inhibition and Medicinal Chemistry (year: 2016, volume: 31, pages: 14–22), Publisher: Taylor & Francis
    Status:
    Published
    DOI:
    10.3109/14756366.2014.1003214 – link to the publication

  10. Antimicrobial and physicochemical characterizations of thiosemicarbazide and s-triazole derivatives

    Authors:
    Edyta Kuśmierz, Agata Siwek, Urszula Kosikowska, Anna Malm, Tomasz Plech, Andrzej Wróbel, Monika Wujec 
    Academic press:
    Phosphorus, Sulfur, and Silicon and the Related Elements (year: 2014, volume: 189, pages: 46029), Publisher: Taylor & Francis
    Status:
    Published
    DOI:
    10.1080/10426507.2014.902831 – link to the publication

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Graphic design and implementation: Jakub Piotrowski