Diversity-Oriented Synthesis of alkaloid-like piperidines as novel privileged structures of potential drugs
2016/23/N/ST5/00101
Keywords
Descriptors
- ST5_23: Chemia organiczna
- ST5_16: Chemia biologiczna
- ST4_11: Nowoczesne metody prowadzenia reakcji i procesów
Panel
ST5 – Materials: materials synthesis, structure-properties relations, advanced and functional materials with designed properties, (macro)molecular architecture, material engineering
Host institution
Zachodniopomorski Uniwersytet Technologiczny w Szczecinie, Wydział Technologii i Inżynierii Chemicznej
Voivodeship: zachodniopomorskie
Principal investigator (from the host institution)
Number of co-investigators in the project: 3
Call
PRELUDIUM 12 – announced on 2016-09-15
- Amount awarded
- 150 000 PLN
- Project start date
- 2017-07-20
- Project end date
- 2020-07-19
- Project duration
- 36 months (the same as in the proposal)
- Project status
- Project settled
Project description
Download the project description in a pdf file
Note — project descriptions were prepared by the authors of the applications themselves and placed in the system in an unchanged form.
Equipment purchased [PL]
- Membranowa pompa próżniowa. Cost: 3 500 PLN
- Mieszadło magnetyczne. Cost: 3 000 PLN
- Wyparka obrotowa. Cost: 13 900 PLN
Information in the final report
Publication in academic press/journals (4)
-
Diversity-Oriented Synthesis toward Fused and Bridged Benzobicyclic Piperidin(on)es
- Authors:
- Tomasz J. Idzik, Zofia M. Myk, Jacek G. Sośnicki
- Academic press:
- Journal of Organic Chemistry (year: 2019, volume: 84, pages: 8046−8066), Publisher: American Chemical Society
- Status:
- Published
- DOI:
- 10.1021/acs.joc.9b00920 – link to the publication
-
Synthesis of Polycyclic δ-Lactams with Bridged Benzomorphan Skeleton: Selectivity and Diversity Driven by Substituents
- Authors:
- Jacek G. Sośnicki, Tomasz J. Idzik, Aleksandra Borzyszkowska, Gabriela Maciejewska, Łukasz Struk
- Academic press:
- The Journal of Organic Chemistry (year: 2018, volume: 83, pages: 1745-1760), Publisher: American Chemical Society
- Status:
- Published
- DOI:
- 10.1021/acs.joc.7b02509 – link to the publication
-
Magnesiate-Utilized/Benzyne-Mediated Approach to Indenopyridones from 2‑Pyridones: An Attempt To Synthesize the Indenopyridine Core of Haouamine
- Authors:
- Tomasz J. Idzik, Aleksandra Borzyszkowska-Ledwig, Łukasz Struk, Jacek G. Sośnicki
- Academic press:
- Organic Letters (year: 2019, volume: 21, pages: 9667−9671), Publisher: American Chemical Society
- Status:
- Published
- DOI:
- 10.1021/acs.orglett.9b03806 – link to the publication
-
Pyridones – Powerful Precursors for the Synthesis of Alkaloids, Their Derivatives, and Alkaloid-Inspired Compounds
- Authors:
- Jacek G. Sośnicki, Tomasz J. Idzik
- Academic press:
- Synthesis (year: 2019, volume: 51, pages: 3369–3396), Publisher: Thieme Chemistry
- Status:
- Published
- DOI:
- 10.1055/s-0037-1611844 – link to the publication